Reductive Heck reactions of N-arylamino-substituted tricyclic imides

Main Article Content

Muge Atbakar
Onur Topbaştekin
Nuket Ocal

Abstract

The C–C coupling of (3aR,4S,7R,7aS)-rel-2-[(3-chloro-4-fluoro­phe­nyl)amino]-3a,4,7,7a-tetrahydro-4,7-methano-1H-isoindole-1,3(2H)-dione (3) which was prepared as a new starting material and (3aR,4S,7R,7aS)-rel-2-[(2,4--dinitrophe­nyl)amino]-3a,4,7,7a-tetrahydro-4,7-methano-1H-isoindole-1,3­(2H)-dione (6) with aryl- and heteroaryl iodides gave the aryl(hetaryl), N-aryl­amino tricyclic imides 4ad and 7ad under reductive Heck conditions.

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How to Cite
[1]
M. Atbakar, O. Topbaştekin, and N. Ocal, “Reductive Heck reactions of N-arylamino-substituted tricyclic imides”, J. Serb. Chem. Soc., vol. 81, no. 10, pp. 1121–1125, Oct. 2016.
Section
Organic Chemistry
Author Biographies

Muge Atbakar, Yildiz Technical University, Faculty of Science and Arts, Department of Chemistry, Davutpasa Campus, 34220, Esenler-Istanbul

Chemistry

Onur Topbaştekin, Yildiz Technical University, Faculty of Science and Arts, Department of Chemistry, Davutpasa Campus, 34220, Esenler-Istanbul

Chemistry

 

 

 

Nuket Ocal, Yildiz Technical University, Faculty of Science and Arts, Department of Chemistry, Davutpasa Campus, 34220, Esenler-Istanbul

Chemistry

References

S. Tsupova, U. Maeorg, Heterocycles 88 (2014) 129

Z. Cui, X. Yang, Y. Shi, H. Uzawa, J. Cui, Bioorg. Med. Chem. Lett. 21 (2011) 7193

O. V. Krishchik, I. N. Tarabara, A. O. Kasyan, S. V. Shishkina, O. V. Shishkin, A. K. Isaev, L. I. Kasyan, Russ. J. Org. Chem. 40 (2004) 1140

M. F. Brana, A. Gradillas, A. Gomez, N. Acero, F. Llinares, D. Munoz-Mingarrro, C. Abradelo, F. Rey-Stolle, M. Yuste, J. Campos, M. A. Gallo, A. Espinosa, J. Med. Chem. 47 (2004) 2236

S. M. Sondhi, R. Rani, P. Roy, S. K. Agrawal, A. K. Saxena, Bioorg. Med. Chem. Lett. 19 (2009) 1534

J. Kossakowski, M. Jarocka, Farmaco 56 (2001) 785

M. M. Patil, S. S. Rajput, Int. J. Pharm. Pharm. Sci. 6 (2014) 8

M. K. Hargreaves, J. G. Pritchard, H. R. Dave, Chem. Rev. 70 (1970) 439

E. Negishi, A. Meijere, Handbook of organopalladium chemistry for organic synthesis, Wiley, New York, 2002, p. 1113

I. P. Beletskaya, A. V. Cheprakov, Chem. Rev. 100 (2000) 3009

Z. L. Wei, C. George, A. P. Kozikowski, Tetrahedron Lett. 44 (2003) 3847

J. Storsberg, M.-L. Yao, N. Ocal, A. de Meijere, A. E. W. Adam, D. E. Kaufmann, Chem. Commun. (2005) 5665

C. Yolacan, E. Bagdatli, N. Ocal, D. E. Kaufmann, Helv. Chim. Acta 90 (2007) 2380

G. Goksu, M. Gul, N. Ocal, D. E. Kaufmann, Tetrahedron Lett. 49 (2008) 2685

C. Celik, I. Kulu, N. Ocal, D. E. Kaufmann, Helv. Chim. Acta 92 (2009) 1092

G. Goksu, N. Ocal D. E. Kaufmann, Molecules 15 (2010) 1302

J. C. Namyslo, J. Storsberg, J. Klinge, C. Gartner, M. Yao, N. Ocal, D. E. Kaufmann, Molecules 15 (2010) 3402

M. Gul, I. Kulu, N. Ocal, J. Chem. Res. 37 (2013) 345

J. C. Namyslo, D. E. Kaufmann, Chem. Ber./Recl. 130 (1997) 1327

F. Stuhlmann, D. E. Kaufmann, J. Prakt. Chem. 341 (1999) 455

J. C. Namyslo, D. E. Kaufmann, Synlett 6 (1999) 804

K. K. W. To, X. Wang, C. W. Yu, Y.-P. Ho, S. C. F. Au-Yeung, Bioorg. Med. Chem. 12 (2004) 4565.